Tarzia, Giorgio: шукати на сайті Z-Library

Giorgi, Luca, Piersanti, Giovanni, Bartoccini, Francesca, Tarzia, Giorgio, Minetti, Patrizia, Gallo, Grazia, Giorgi, Fabrizio, Castorina, Massimo, Ghirardi, Orlando, Carminati, Paolo

Рік:

2009

Мова:

english

Файл:

PDF, 271 KB

english, 2009

Synthesis of benzo[1,2-d;3,4-d′]diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists

Журнал:

Organic & Biomolecular Chemistry

Рік:

2007

Мова:

english

Файл:

PDF, 146 KB

english, 2007

Pyrrolopyridine analogs of nalidixic acid. 1. Pyrrolo[2,3-b]pyridines

Emilio Toja, Giorgio Tarzia, Pietro Ferrari, Giorgio Tuan

Журнал:

Journal of Heterocyclic Chemistry

Рік:

1986

Мова:

english

Файл:

PDF, 470 KB

english, 1986

Conformationally Restrained Melatonin Analogues: Synthesis, Binding Affinity for the Melatonin Receptor, Evaluation of the Biological Activity, and Molecular Modeling Study

Spadoni, Gilberto, Balsamini, Cesarino, Diamantini, Giuseppe, Di Giacomo, Barbara, Tarzia, Giorgio, Mor, Marco, Plazzi, Pier Vincenzo, Rivara, Silvia, Lucini, Valeria, Nonno, Romolo, Pannacci, Marilou

Журнал:

Journal of Medicinal Chemistry

Рік:

1997

Мова:

english

Файл:

PDF, 510 KB

english, 1997

Letter to the Editor: Correlation of the mutagenic properties of aryl- and heteroaryltriazenes with their electron ionization induced fragmentation

Giorgio Tarzia, G. Diamantini, Andrea Tontini, Donato Favretto, Pietro Traldi

Журнал:

Rapid Communications in Mass Spectrometry

Рік:

1996

Мова:

english

Файл:

PDF, 301 KB

english, 1996

Correlation of the antimetastatic properties of aryltriazenes with their electron impact ionization mass spectrometry

Giorgio Tarzia, Giuseppe Diamantini, Andrea Tontini, Annalida Bedini, Donata Favretto, Pietro Traldi

Журнал:

Rapid Communications in Mass Spectrometry

Рік:

1997

Мова:

english

Файл:

PDF, 83 KB

english, 1997

Synthesis and Evaluation of 1,5-Benzodiazepines with Bridged Cycloalkyl Substituents at the N-1 Position as Potent and Selective CCK-B Ligands

Gabriella Finizia, Daniele Donati, Giorgio Pentassuglia, Stefano Polinelli, Giorgio Tarzia, Maria Elvira Tranquillini, Antonella Ursini

Журнал:

Archiv der Pharmazie

Рік:

1998

Мова:

english

Файл:

PDF, 66 KB

english, 1998

Identification of a Bioactive Impurity in a Commercial Sample of 6-Methyl-2-p-Tolylaminobenzo[d][1,3]Oxazin-4-One (URB754)

Giorgio Tarzia, Francesca Antonietti, Andrea Duranti, Andrea Tontini, Marco Mor, Silvia Rivara, Pietro Traldi, Giuseppe Astarita, Alvin King, Jason R. Clapper, Daniele Piomelli

Журнал:

Annali di Chimica

Рік:

2007

Мова:

english

Файл:

PDF, 248 KB

english, 2007

Novel 1,5-Benzodiazepines as CCK-B Ligands. Effect of Aryl-Carbamic Substituents at the C-3 Position Together with Halogen Substitution on the Benzo-Fused Ring

M. Elvira Tranquillini, Paolo G. Cassarà, Mauro Corsi, Giovanni Curotto, Daniele Donati, Gabriella Finizia, Giorgio Pentassuglia, Stefano Polinelli, Giorgio Tarzia, Antonella Ursini, Franciscus T. M.

Журнал:

Archiv der Pharmazie

Рік:

1997

Мова:

english

Файл:

PDF, 532 KB

english, 1997

Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors

Marco Mor, Silvia Rivara, Alessio Lodola, Simone Lorenzi, Fabrizio Bordi, Pier Vincenzo Plazzi, Gilberto Spadoni, Annalida Bedini, Andrea Duranti, Andrea Tontini, Giorgio Tarzia

Журнал:

Chemistry & Biodiversity

Рік:

2005

Мова:

english

Файл:

PDF, 425 KB

english, 2005

ChemInform Abstract: Rotation about the N2—N3 Bond in 3,3-Dimethyl-1-(isoxazol-3-yl)-triazenes.

Andrea Tontini, Giuseppe Gatti, Giuseppe Diamantini, Giorgio Tarzia

Журнал:

Рік:

1999

Файл:

PDF, 29 KB

1999

ChemInform Abstract: 3-(2-Carbamoylvinyl)-4,5-dimethylpyrrole-2-carboxylic Acids as Ligands at the NMDA Glycine-Binding Site: A Study on the 2-Carbamoylvinyl Chain Modification.

Cesarino Balsamini, Annalida Bedini, Giuseppe Diamantini, Gilberto Spadoni, Giorgio Tarzia, Andrea Tontini, Romano Di Fabio, Daniele Donati

Журнал:

Giorgio Tarzia, Giuseppe Diamantini, Marco Mor, Gilberto Spadoni

Рік:

1999

Файл:

PDF, 31 KB

1999

ChemInform Abstract: Design and Synthesis of Melatonin Receptors Agonists and Antagonists

Журнал:

Рік:

2000

Файл:

PDF, 24 KB

2000

ChemInform Abstract: Synthesis and Characterization of a Peripherally Restricted CB1 Cannabinoid Antagonist, URB447, that Reduces Feeding and Body-Weight Gain in Mice.

Jesse LoVerme, Andrea Duranti, Andrea Tontini, Gilberto Spadoni, Marco Mor, Silvia Rivara, Nephi Stella, Cong Xu, Giorgio Tarzia, Daniele Piomelli

Журнал:

Francesca Bartoccini, Walter Cabri, Diana Celona, Patrizia Minetti, Giovanni Piersanti, Giorgio Tarzia

Рік:

2009

Файл:

PDF, 23 KB

2009

ChemInform Abstract: Direct B-Alkyl Suzuki—Miyaura Cross-Coupling of 2-Halopurines. Practical Synthesis of ST1535 (VII), a Potent Adenosine A2A Receptor Antagonist.

Журнал:

Рік:

2010

Файл:

PDF, 31 KB

2010

Synthesis and Structure–Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring

Giorgio Tarzia, Andrea Duranti, Giuseppe Gatti, Giovanni Piersanti, Andrea Tontini, Silvia Rivara, Alessio Lodola, Pier Vincenzo Plazzi, Marco Mor, Satish Kathuria, Daniele Piomelli

Журнал:

Rainer Metternich, Giorgio Tarzia, Guiseppe Ronsisvalle, Hans Ulrich Stilz

Рік:

2006

Мова:

english

Файл:

PDF, 354 KB

english, 2006

The Pipeline Is Filled…

Журнал:

Рік:

2006

Мова:

english

Файл:

PDF, 405 KB

english, 2006

Drug Discovery Handbook. Edited by Shayne Cox Gad.

Giorgio Tarzia

Журнал:

Рік:

2006

Мова:

english

Файл:

PDF, 34 KB

english, 2006

Towards the Development of Mixed MT1-Agonist/MT2-Antagonist Melatonin Receptor Ligands

Gilberto Spadoni, Annalida Bedini, Tomaso Guidi, Giorgio Tarzia, Valeria Lucini, Marilou Pannacci, Franco Fraschini

Журнал:

Рік:

2006

Мова:

english

Файл:

PDF, 139 KB

english, 2006

Synthesis, Enantiomeric Resolution, and Structure–Activity Relationship Study of a Series of 10,11-Dihydro-5H-Dibenzo[a,d]cycloheptene MT2 Receptor Antagonists

Gilberto Spadoni, Annalida Bedini, Giuseppe Diamantini, Giorgio Tarzia, Silvia Rivara, Simone Lorenzi, Alessio Lodola, Marco Mor, Valeria Lucini, Marilou Pannacci, Alessia Caronno, Franco Fraschini

Журнал:

Rainer Metternich, Giorgio Tarzia

Рік:

2007

Мова:

english

Файл:

PDF, 391 KB

english, 2007

Medicinal Chemistry: Defining Itself

Журнал:

Рік:

2008

Мова:

english

Файл:

PDF, 245 KB

english, 2008

A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo

Jason R. Clapper, Federica Vacondio, Alvin R. King, Andrea Duranti, Andrea Tontini, Claudia Silva, Silvano Sanchini, Giorgio Tarzia, Marco Mor, Daniele Piomelli

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 302 KB

english, 2009

Cover Picture: Structure–Property Relationships of a Class of Carbamate-Based Fatty Acid Amide Hydrolase (FAAH) Inhibitors: Chemical and Biological Stability / A Second Generation of Carbamate-Based Fatty Acid Amide Hydrolase Inhibitors with Improved Activity in vivo (ChemMedChem 9/2009)

Federica Vacondio, Claudia Silva, Alessio Lodola, Alessandro Fioni, Silvia Rivara, Andrea Duranti, Andrea Tontini, Silvano Sanchini, Jason R. Clapper, Daniele Piomelli, Marco Mor, Giorgio Tarzia, Alvi

Журнал:

Rainer Metternich, Giorgio Tarzia

Рік:

2009

Мова:

english

Файл:

PDF, 792 KB

english, 2009

“Hot Spots” in Medicinal Chemistry

Журнал:

Рік:

2010

Мова:

english

Файл:

PDF, 285 KB

english, 2010

Electron impact ionization and fast atom bombardment mass spectrometry of some 3,3-dimethyl-1-(isoxazol-3-yl)triazenes, a new class of potential anticancer agents

Laura Orsatti, Roberta Seraglia, Pietro Traldi, Giuseppe Diamantini, Giorgio Tarzia, Andrea Tontini

Журнал:

Рік:

1995

Мова:

english

Файл:

PDF, 423 KB

english, 1995

Correlation between energetics of collisionally activated decompositions, interaction energy and biological potency of carbamate FAAH inhibitors

Giovanni Valitutti, Andrea Duranti, Alessio Lodola, Marco Mor, Giovanni Piersanti, Daniele Piomelli, Silvia Rivara, Andrea Tontini, Giorgio Tarzia, Pietro Traldi

Журнал:

Рік:

2007

Мова:

english

Файл:

PDF, 111 KB

english, 2007

The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity

Giovanni Valitutti, Andrea Duranti, Marco Mor, Giovanni Piersanti, Daniele Piomelli, Silvia Rivara, Andrea Tontini, Giorgio Tarzia, Pietro Traldi

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 100 KB

english, 2009

Erratum: The collisional behavior of ESI-generated protonated molecules of some carbamate FAAH inhibitors isosteres and its relationships with biological activity

Giovanni Valitutti, Andrea Duranti, Marco Mor., Giovanni Piersanti, Daniele Piomelli, Silvia Rivara, Andrea Tontini, Giorgio Tarzia, Pietro Traldi

Журнал:

Рік:

2011

Файл:

PDF, 28 KB

2011

Tandem mass spectrometric data–FAAH inhibitory activity relationships of some carbamic acid O-aryl esters

Elisa Basso, Andrea Duranti, Marco Mor, Daniele Piomelli, Andrea Tontini, Giorgio Tarzia, Pietro Traldi

Журнал:

Mahmoud Hamdan, Giorgio Tarzia, Cesarino Balsamini, Gilberto Spadoni, Ornella Curcuruto, Pietro Traldi

Рік:

2004

Мова:

english

Файл:

PDF, 172 KB

english, 2004

Positive-ion mass spectra and collision-induced dissociation of some 2,3-didehydro amino acids

Журнал:

Bahman M. Sadeghpouiy, Roberto Pellicciari, Carla Marchioro, Tino Rossi, Bruno Tamburini, Giorgio Tarzia, Antonella Ursini

Рік:

1990

Мова:

english

Файл:

PDF, 590 KB

english, 1990

Synthesis of 6α-methoxy-6β-hydroxymethylpenems

Журнал:

Tetrahedron

Рік:

1995

Мова:

english

Файл:

PDF, 593 KB

english, 1995

Anti-hypertensives: 1-alkyl-2-arylpiperazinoethyl-1H-naphth[1,2-d]imidazoles

Emilio Toja, Giuseppe Di Francesco, Domenico Barone, Emiliana Baldoli, Nerina Corsico, Giorgio Tarzia

Журнал:

European Journal of Medicinal Chemistry

Рік:

1987

Мова:

english

Файл:

PDF, 992 KB

english, 1987

Reassessing the melatonin pharmacophore—Enantiomeric resolution, pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue

Silvia Rivara, Giuseppe Diamantini, Barbara Di Giacomo, Doriano Lamba, Giuseppe Gatti, Valeria Lucini, Marilou Pannacci, Marco Mor, Gilberto Spadoni, Giorgio Tarzia

Журнал:

Barbara Di Giacomo, Annalida Bedini, Gilberto Spadoni, Giorgio Tarzia, Franco Fraschini, Marilou Pannacci, Valeria Lucini

Рік:

2006

Мова:

english

Файл:

PDF, 301 KB

english, 2006

Synthesis and biological activity of new melatonin dimeric derivatives

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2007

Мова:

english

Файл:

PDF, 187 KB

english, 2007

Synthesis and characterization of a peripherally restricted CB1 cannabinoid antagonist, URB447, that reduces feeding and body-weight gain in mice

Jesse LoVerme, Andrea Duranti, Andrea Tontini, Gilberto Spadoni, Marco Mor, Silvia Rivara, Nephi Stella, Cong Xu, Giorgio Tarzia, Daniele Piomelli

Журнал:

Рік:

2009

Мова:

english

Файл:

PDF, 478 KB

english, 2009

URB602 Inhibits Monoacylglycerol Lipase and Selectively Blocks 2-Arachidonoylglycerol Degradation in Intact Brain Slices

Alvin R. King, Andrea Duranti, Andrea Tontini, Silvia Rivara, Anja Rosengarth, Jason R. Clapper, Giuseppe Astarita, Jennifer A. Geaga, Hartmut Luecke, Marco Mor, Giorgio Tarzia, Daniele Piomelli

Журнал:

Chemistry & Biology

Рік:

2007

Мова:

english

Файл:

PDF, 342 KB

english, 2007

Reactions of 3-carbomethoxy-2-aza-1,3-butadiene derivatives with dienophiles

Cesarino Balsamini, Annalida Bedini, Roberta Galarini, Gilberto Spadoni, Giorgio Tarzia, Mahmoud Hamdan

Журнал:

Tetrahedron

Рік:

1994

Мова:

english

Файл:

PDF, 1.23 MB

english, 1994

University education of medicinal chemists: comparison of eight countries

C.Robin Ganellin, Lester A Mitscher, Bernd Clement, Toshi-Hiko Kobayashi, Emilio Kyburz, Olivier Lafont, Annie Marcincal, Antonio Monge, Giorgio Tarzia, John G Topliss

Журнал:

European Journal of Medicinal Chemistry

Рік:

2000

Мова:

english

Файл:

PDF, 62 KB

english, 2000

2,4-Dicarboxy-pyrroles as selective non-Competitive mGluR1 antagonists: further characterization of 3,5-Dimethyl pyrrole-2,4-dicarboxylic acid 2-propyl ester 4-(1,2,2-Trimethyl-propyl) ester and structure–Activity relationships

Fabrizio Micheli, Romano Di Fabio, Fabio Bordi, Palmina Cavallini, Paolo Cavanni, Daniele Donati, Stefania Faedo, Micaela Maffeis, Fabio Maria Sabbatini, Giorgio Tarzia, Maria Elvira Tranquillini

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

2003

Мова:

english

Файл:

PDF, 228 KB

english, 2003

Synthesis, antimicrobial activity and binding properties of calix[4]arene based vancomycin mimics

Alessandro Casnati, Massimo Fabbi, Nicola Pelizzi, Andrea Pochini, Francesco Sansone, Rocco Unguro, Enza Di Modugno, Giorgio Tarzia

Журнал:

Bioorganic & Medicinal Chemistry Letters

Рік:

1996

Мова:

english

Файл:

PDF, 309 KB

english, 1996

Synthesis, pharmacological characterization and QSAR studies on 2-substituted indole melatonin receptor ligands

Marco Mor, Gilberto Spadoni, Barbara Di Giacomo, Giuseppe Diamantini, Annalida Bedini, Giorgio Tarzia, Pier Vincenzo Plazzi, Silvia Rivara, Romolo Nonno, Valeria Lucini, Marilou Pannacci, Franco Frasc

Журнал:

Journal of Pineal Research

Рік:

2001

Мова:

english

Файл:

PDF, 337 KB

english, 2001

A new melatonin receptor ligand with mt1-agonist and MT2-antagonist properties

Romolo Nonno, Valeria Lucini, Gilberto Spadoni, Marilou Pannacci, Assunta Croce, Daniele Esposti, Cesarino Balsamini, Giorgio Tarzia, Franco Fraschini, Bojidar M. Stankov

Журнал:

Рік:

2000

Мова:

english

Файл:

PDF, 139 KB

english, 2000

Indole-based analogs of melatonin: in vitro antioxidant and cytoprotective activities

Marco Mor, Claudia Silva, Federica Vacondio, Pier Vincenzo Plazzi, Simona Bertoni, Gilberto Spadoni, Giuseppe Diamantini, Annalida Bedini, Giorgio Tarzia, Morena Zusso, Davide Franceschini, Pietro Giu

Журнал:

Journal of Pineal Research

Рік:

2004

Мова:

english

Файл:

PDF, 179 KB

english, 2004

On the formation of [H3CSSCH3]+. ions from the bis(dimethylthio)mercury molecular ion

Loris Tonidandel, Giorgio Tarzia, Francesca Antonietti, Andrea Vittadini, Pietro Traldi

Журнал:

Rapid Communications in Mass Spectrometry

Рік:

2006

Мова:

english

Файл:

PDF, 174 KB

english, 2006

Hereditary spherocytosis and elliptocytosis associated with prosthetic heart valve replacement: rheological study of erythrocyte modifications

Patrizia Caprari, Anna Tarzia, Giorgio Mojoli, Paolo Cianciulli, Emilio Mannella, Maria Cristina Martorana

Журнал:

International Journal of Hematology

Рік:

2009

Мова:

english

Файл:

PDF, 364 KB

english, 2009

Synthesis of 6β-methoxy-6α-hydroxymethylpenems

Bahman M. Sadeghpour, Roberto Pellicciari, Carla Marchioro, Tino Rossi, Bruno Tamburini, Giorgio Tarzia

Журнал:

Tetrahedron

Рік:

1995

Мова:

english

Файл:

PDF, 552 KB

english, 1995

Bivalent ligand approach on N-{2-[(3-methoxyphenyl)methylamino]ethyl}acetamide: Synthesis, binding affinity and intrinsic activity for MT1 and MT2 melatonin receptors

Gilberto Spadoni, Annalida Bedini, Pierfrancesco Orlando, Simone Lucarini, Giorgio Tarzia, Marco Mor, Silvia Rivara, Valeria Lucini, Marilou Pannacci, Francesco Scaglione

Журнал:

Рік:

2011

Мова:

english

Файл:

PDF, 444 KB

english, 2011

Synthesis and structure–activity relationships of a series of pyrrole cannabinoid receptor agonists

Giorgio Tarzia, Andrea Duranti, Andrea Tontini, Gilberto Spadoni, Marco Mor, Silvia Rivara, Pier Vincenzo Plazzi, Satish Kathuria, Daniele Piomelli

Журнал: